Data | Título | Autor(es) | Tipo | Acesso |
2020 | 4,9‐Diaminoacridines and 4‐Aminoacridines as dual‐stage antiplasmodial hits | Fonte, Mélanie; Tassi, Natália; Fontinha, Diana; Bouzón‐Arnáiz, Inés; Ferraz, Ricardo; Araújo, Maria J.; Fernàndez‐Busquets, Xavier; Prudêncio, Miguel; Gomes, Paula; Teixeira, Cátia | article |  |
2008 | Amino acids as selective acylating agents | Vale, Nuno; Matos, Joana; Moreira, Rui; Gomes, Paula | article |  |
2009 | Anti-tumoral activity of imidazoquines, a new class of antimalarials derived from primaquine | Fernandes, Iva; Vale, Nuno; de Freitas, Victor; Moreira, Rui; Mateus, Nuno; Gomes, Paula | article |  |
2008 | Characterization of primaquine imidazolidin-4-ones with antimalarial activity by electrospray ionization-ion trap mass spectrometry | Vale, Nuno; Moreira, Rui; Gomes, Paula | article |  |
2019 | Cinnamic acid conjugates in the rescuing and repurposing of classical antimalarial drugs | Silva, Ana Teresa; Bento, Clara M.; Pena, Ana C; Figueiredo, Luisa M.; Prudêncio, Cristina; Aguiar, Luísa; Silva, Tânia; Ferraz, Ricardo; Gomes, Maria Salomé; Teixeira, Cátia; Gomes, Paula | article |  |
2019 | Coupling the cell-penetrating peptides transportan and transportan 10 to primaquine enhances its activity against liver-stage malaria parasites | Aguiar, Luísa; Machado, Marta; Sanches-Vaz, Margarida; Prudêncio, Miguel; Vale, Nuno; Gomes, Paula | article |  |
2007 | Cyclization-activated prodrugs | Gomes, Paula; Vale, Nuno; Moreira, Rui | article |  |
2008 | Dipeptide derivatives of AZT | Santos, Cledir; Morais, Jose; Gouveia, Luis; de Clercq, Erik; Pannecouque, Christophe; Nielsen, Carsten Uhd; Steffansen, Bente; Moreira, Rui; Gomes, Paula | article |  |
2009 | Electrospray ionization mass spectrometry as a valuable tool in the characterization of novel primaquine peptidomimetic derivatives | Vale, Nuno; Matos, Joana; Moreira, Rui; Gomes, Paula | article |  |
2008 | Electrospray Ionization-Ion Trap Mass Spectrometry Study of PQAAPro and PQProAA Mimetic Derivatives of the Antimalarial Primaquine | Vale, Nuno; Matos, Joana; Moreira, Rui; Gomes, Paula | article |  |
2008 | Imidazolidin-4-one peptidomimetic derivatives of primaquine | Vale, Nuno; Matos, Joana; Gut, Jiri; Nogueira, Fatima; do Rosario, Virgilio; Rosenthal, Philip J.; Moreira, Rui; Gomes, Paula | article |  |
2009 | Imidazoquines as Antimalarial and Antipneumocystis Agents | Vale, Nuno; Prudencio, Miguel; Marques, Catarina A.; Collins, Margaret S.; Gut, Jiri; Nogueira, Fatima; Matos, Joana; Rosenthal, Philip J.; Cushion, Melanie T.; do Rosario, Virgilio E.; Mota, Maria M.; Moreira, Rui; Gomes, Paula | article |  |
2022 | Neuroprotective effects on microglia and insights into the structure–activity relationship of an antioxidant peptide isolated from Pelophylax perezi | Plácido, Alexandra; Amaral, Constança Pais Do; Teixeira, Cátia; Nogueira, Ariane; Brango‐Vanegas, José; Alves Barbosa, Eder; C. Moreira, Daniel; Silva‐Carvalho, Amandda E.; da Silva, Maria da Gloria; do Nascimento Dias, Jhones; Albuquerque, Patrícia; Saldanha‐Araújo, Felipe; C. D. A. Lima, Filipe; Batagin‐Neto, Augusto; Kuckelhaus, Selma; Bessa, Lucinda J.; Freitas, Jaime; Dotto Brand, Guilherme; Santos, Nuno C.; B. Relvas, João; Gomes, Paula; S. A. Leite, José Roberto; Eaton, Peter | article |  |
2023 | New 4-(N-cinnamoylbutyl)aminoacridines as potential multi-stage antiplasmodial leads | Fonte, Mélanie; Fontinha, Diana; Moita, Diana; Caño-Prades, Omar; Avalos-Padilla, Yunuen; Fernàndez-Busquets, Xavier; Prudêncio, Miguel; Gomes, Paula; Teixeira, Cátia | article |  |
2009 | Primaquine dipeptide derivatives bearing an imidazolidin-4-one moiety at the N-terminus as potential antimalarial prodrugs | Vale, Nuno; Nogueira, Fatima; do Rosario, Virgilio E.; Gomes, Paula; Moreira, Rui | article |  |
2006 | Reactivity of imidazolidin-4-one derivatives of primaquine | Chambel, Paula; Capela, Rita; Lopes, Francisca; Iley, Jim; Morais, Jose; Gouveia, Luis; Gomes, Jose R. B.; Gomes, Paula; Moreira, Rui | article |  |
2009 | Structure-activity relationships for dipeptide prodrugs of acyclovir | Santos, Cledir R.; Capela, Rita; Pereira, Claudia S. G. P.; Valente, Emilia; Gouveia, Luis; Pannecouque, Christophe; De Clercq, Erik; Moreira, Rui; Gomes, Paula | article |  |
2009 | TOWARDS DUAL-ACTION ANTI-MALARIALS - PRIMACENES, FERROCENE DERIVATIVES OF PRIMAQUINE | Matos, Joana; Vale, Nuno; Moreira, Rui; Gomes, Paula | article |  |
2007 | Unanticipated stereoselectivity in the reaction of primaquine alpha-aminoamides with substituted benzaldehydes | Ferraz, Ricardo; Gomes, Jose R. B.; de Oliveira, Eliandre; Moreira, Rui; Gomes, Paula | article |  |
2006 | Waste treatment by an Incinerator : what about health-related quality of life? | Reis, Maria de Fátima; Santos, Osvaldo; Gomes, Paula; Aniceto, Pedro; Aguiar, Pedro; Melim, Maurício; Cardoso, Liliana; Pereira Miguel, José | conferenceObject |  |